阿西替尼是一种 VEGFR 抑制剂,高浓度时也抑制 PDGFR,作用于 VEGFR1,VEGFR2,VEGFR3 和 PDGFRβ,IC50 分别为 0.1 nM,0.2 nM,0.1-0.3 nM 和 1.6 nM,是一种小分子酪氨酸激酶抑制剂。

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886230-77-9
(E)-6-Iodo-3-(2-(pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
(E)-6-Iodo-3-(2-(pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
品牌:毕得
BD632939886230-77-998%
登录 5g 常备现货
885126-34-1
2-((3-Iodo-1H-indazol-6-yl)thio)-N-methylbenzamide
2-((3-Iodo-1H-indazol-6-yl)thio)-N-methylbenzamide
品牌:毕得
BD235568885126-34-198+%
登录 1g 常备现货
20054-45-9
2-Mercapto-N-methylbenzamide
2-Mercapto-N-methylbenzamide
品牌:毕得
BD16864120054-45-998%
登录 1g 常备现货
261953-36-0
6-Iodo-1H-indazole
6-Iodo-1H-indazole
品牌:毕得
BD28210261953-36-098%
登录 100g 常备现货
70315-70-7
3-Iodo-6-nitro-1H-indazole
3-Iodo-6-nitro-1H-indazole
品牌:毕得
BD8749670315-70-797%
登录 25g 常备现货
319460-85-0
(E)-N-Methyl-2-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)benzamide
(E)-N-Methyl-2-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)benzamide
品牌:毕得
BD114869319460-85-098%
登录 100mg 常备现货
115666-47-2
6-Iodo-1H-indole
6-Iodo-1H-indole
品牌:毕得
BD173568115666-47-297%
登录 10g 常备现货
4363-35-3
(Z/E)-Styrylboronic acid
(Z/E)-Styrylboronic acid
品牌:毕得
BD2231754363-35-395%
登录 5g 常备现货
7597-18-4
6-Nitro-1H-indazole
6-Nitro-1H-indazole
品牌:毕得
BD225137597-18-495%
登录 25g 常备现货
885126-35-2
N-Methyl-2-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-6-yl]thio]benzamide
N-Methyl-2-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-6-yl]thio]benzamide
品牌:毕得
BD00796566885126-35-297%
登录 100mg 常备现货
73870-22-1
Triphenyl(pyridin-2-ylmethyl)phosphonium bromide
Triphenyl(pyridin-2-ylmethyl)phosphonium bromide
品牌:毕得
BD0095187573870-22-198%
登录 1g 常备现货
885518-80-9
6-Iodo-1H-indazole-3-carbaldehyde
6-Iodo-1H-indazole-3-carbaldehyde
品牌:毕得
BD447614885518-80-998%
登录 250mg
944835-85-2
2-((1H-Indazol-6-yl)thio)-N-methylbenzamide
2-((1H-Indazol-6-yl)thio)-N-methylbenzamide
品牌:毕得
BD450031944835-85-295%
登录 250mg
886230-76-8
(E)-3-(2-(Pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-6-amine
(E)-3-(2-(Pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-6-amine
品牌:毕得
BD636768886230-76-897% mix TBC as stabilizer
登录 250mg
886230-74-6
3-Iodo-6-nitro-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
3-Iodo-6-nitro-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
品牌:毕得
BD245057886230-74-695+%
登录 1g
886230-75-7
(E)-6-Nitro-3-(2-(pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
(E)-6-Nitro-3-(2-(pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
品牌:毕得
BD245059886230-75-795% mix TBC as stabilizer
登录 1g
319472-83-8
1H-indazole, 3-iodo-6-nitro-1-[[2-(trimethylsilyl)ethoxy]methyl]-
1H-indazole, 3-iodo-6-nitro-1-[[2-(trimethylsilyl)ethoxy]methyl]-
品牌:毕得
BD00944630319472-83-895%
登录 1g
38700-15-1
Triphenyl(pyridin-2-ylmethyl)phosphonium chloride
Triphenyl(pyridin-2-ylmethyl)phosphonium chloride
品牌:毕得
BD0092171438700-15-198+%
登录 1g
1