吉尔特利尼是一种有效的 FLT3/AXL受体酪氨酸激酶 抑制剂,IC50 分别为 0.29 nM/0.73 nM。

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1254058-34-8
3-Methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)aniline
3-Methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)aniline
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BD2980871254058-34-897%
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313340-08-8
3,5-Dichloro-6-ethylpyrazine-2-carboxamide
3,5-Dichloro-6-ethylpyrazine-2-carboxamide
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BD284646313340-08-897%
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1254053-84-3
6-Ethyl-3-((3-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)amino)-5-((tetrahydro-2H-pyran-4-yl)amino)pyrazine-2-carboxamide hemifumarate
6-Ethyl-3-((3-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)amino)-5-((tetrahydro-2H-pyran-4-yl)amino)pyrazine-2-carboxamide hemifumarate
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BD007758161254053-84-399%
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