罗拉吡坦是高效选择性具有口服活性的 neurokinin NK1 受体抑制剂,Ki值为0.66 nM,为治疗化疗所致恶心呕吐(CINV)的药物。

清空选项
1214741-21-5
(3R,7aR)-3-(tert-butyl)-1-hydroxy-7a-vinyltetrahydropyrrolo[1,2-c]oxazol-5(3H)-one
(3R,7aR)-3-(tert-butyl)-1-hydroxy-7a-vinyltetrahydropyrrolo[1,2-c]oxazol-5(3H)-one
品牌:毕得
BD4477541214741-21-597%
登录 1g 常备现货
1779-49-3
Methyltriphenylphosphonium bromide
Methyltriphenylphosphonium bromide
品牌:毕得
BD1400041779-49-398%
登录 500g 常备现货
552292-08-7
(5S,8S)-8-(((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-1,7-diazaspiro[4.5]decan-2-one
(5S,8S)-8-(((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-1,7-diazaspiro[4.5]decan-2-one
品牌:毕得
BD755781552292-08-799%
登录 100mg 常备现货
205654-80-4
(2R,4S)-Benzyl 5-oxo-2,4-diphenyloxazolidine-3-carboxylate
(2R,4S)-Benzyl 5-oxo-2,4-diphenyloxazolidine-3-carboxylate
品牌:毕得
BD766678205654-80-498%
登录 25g 常备现货
1214741-20-4
(3R,7AR)-3-(tert-butyl)-7a-vinyldihydropyrrolo[1,2-c]oxazole-1,5(3H,6H)-dione
(3R,7AR)-3-(tert-butyl)-7a-vinyldihydropyrrolo[1,2-c]oxazole-1,5(3H,6H)-dione
品牌:毕得
BD4476901214741-20-495%
登录 1g
75-75-2
Methanesulfonicacid
Methanesulfonicacid
品牌:毕得
BD3484375-75-298%
登录 100mL
530441-95-3
(R)-1-(1-(Bromomethoxy)ethyl)-3,5-bis(trifluoromethyl)benzene
(R)-1-(1-(Bromomethoxy)ethyl)-3,5-bis(trifluoromethyl)benzene
品牌:毕得
BD294822530441-95-395+%
登录 1g
1178515-20-2
(R)-5-((((S)-1-((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)-2-phenylbut-3-en-2-yl)amino)methyl)-5-vinylpyrrolidin-2-one
(R)-5-((((S)-1-((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)-2-phenylbut-3-en-2-yl)amino)methyl)-5-vinylpyrrolidin-2-one
品牌:毕得
BD3331431178515-20-295% mix TBC as stabilizer
登录 1g
914462-92-3
(5S,8S)-8-(((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-1,7-diazaspiro[4.5]decan-2-one hydrochloride hydrate
(5S,8S)-8-(((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-1,7-diazaspiro[4.5]decan-2-one hydrochloride hydrate
品牌:毕得
BD316105914462-92-398%
登录 25mg
171284-84-7
(3R,7aS)-3-(tert-Butyl)dihydropyrrolo[1,2-c]oxazole-1,5(3H,6H)-dione
(3R,7aS)-3-(tert-Butyl)dihydropyrrolo[1,2-c]oxazole-1,5(3H,6H)-dione
品牌:毕得
BD258812171284-84-795%
登录 1g
1214741-14-6
(S)-1-((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)-2-phenylbut-3-en-2-amine fumarate
(S)-1-((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)-2-phenylbut-3-en-2-amine fumarate
品牌:毕得
BD6891531214741-14-697%
登录 250mg
1214741-24-8
(S)-5-((Benzylamino)methyl)pyrrolidin-2-one hydrochloride
(S)-5-((Benzylamino)methyl)pyrrolidin-2-one hydrochloride
品牌:毕得
BD5648581214741-24-895%
登录 250mg
1214741-19-1
(3R,7aR)-3-(tert-Butyl)-1,5-dioxohexahydropyrrolo[1,2-c]oxazole-7a-carbaldehyde
(3R,7aR)-3-(tert-Butyl)-1,5-dioxohexahydropyrrolo[1,2-c]oxazole-7a-carbaldehyde
品牌:毕得
BD7489881214741-19-195%
登录 250mg
530441-36-2
(2R,4S)-Benzyl 4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-5-oxo-2,4-diphenyloxazolidine-3-carboxylate
(2R,4S)-Benzyl 4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-5-oxo-2,4-diphenyloxazolidine-3-carboxylate
品牌:毕得
BD766677530441-36-297%
登录 1g
1214741-17-9
BENZYL ((S)-1-((R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-2-PHENYLBUT-3-EN-2-YL)CARBAMATE
BENZYL ((S)-1-((R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-2-PHENYLBUT-3-EN-2-YL)CARBAMATE
品牌:毕得
BD008721531214741-17-995%
登录 1g
1214741-22-6
(R)-5-Oxo-2-vinylpyrrolidine-2-carbaldehyde
(R)-5-Oxo-2-vinylpyrrolidine-2-carbaldehyde
品牌:毕得
BD013191881214741-22-698% +(stabilized with TBC)
登录 100mg
1