曲美替尼是有效的 MEK 抑制剂,抑制MEK1 和 MEK2的IC50 约为 2 nM。由于Trametinib溶解性差,更加推荐使用 Trametinib DMSO solvate (Cat. No.: HY-10999A)。

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871700-22-0
3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-6-(methylamino)pyrimidine-2,4(1H,3H)-dione
3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-6-(methylamino)pyrimidine-2,4(1H,3H)-dione
品牌:毕得
BD290505871700-22-097%
登录 250mg 常备现货
1187431-43-1
N-(3-(3-Cyclopropyl-5-((2-fluoro-4-iodophenyl)amino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7-tetrahydropyrido[4,3-d]pyrimidin-1(2H)-yl)phenyl)acetamide dimethyl sulfoxide complex
N-(3-(3-Cyclopropyl-5-((2-fluoro-4-iodophenyl)amino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7-tetrahydropyrido[4,3-d]pyrimidin-1(2H)-yl)phenyl)acetamide dimethyl sulfoxide complex
品牌:毕得
BD4482591187431-43-198%
登录 250mg 常备现货
871700-24-2
3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-5-hydroxy-6,8-dimethylpyrido[2,3-d]pyrimidine-2,4,7(1H,3H,8H)-trione
3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-5-hydroxy-6,8-dimethylpyrido[2,3-d]pyrimidine-2,4,7(1H,3H,8H)-trione
品牌:毕得
BD450017871700-24-298%
登录 1g 常备现货
102-28-3
N-(3-Aminophenyl)acetamide
N-(3-Aminophenyl)acetamide
品牌:毕得
BD84390102-28-398%
登录 1kg 常备现货
871700-32-2
3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-6,8-dimethyl-2,4,7-trioxo-1,2,3,4,7,8-hexahydropyrido[2,3-d]pyrimidin-5-yl 4-methylbenzenesulfonate
3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-6,8-dimethyl-2,4,7-trioxo-1,2,3,4,7,8-hexahydropyrido[2,3-d]pyrimidin-5-yl 4-methylbenzenesulfonate
品牌:毕得
BD315971871700-32-298%
登录 1g 常备现货
29632-74-4
2-Fluoro-4-iodoaniline
2-Fluoro-4-iodoaniline
品牌:毕得
BD339829632-74-498%
登录 10g 常备现货
871700-28-6
6-Amino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyrimidine-2,4(1H,3H)-dione
6-Amino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyrimidine-2,4(1H,3H)-dione
品牌:毕得
BD244323871700-28-698%
登录 1g 常备现货
871700-25-3
N-(3-((3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-6,8-dimethyl-2,4,7-trioxo-1,2,3,4,7,8-hexahydropyrido[2,3-d]pyrimidin-5-yl)amino)phenyl)acetamide
N-(3-((3-Cyclopropyl-1-(2-fluoro-4-iodophenyl)-6,8-dimethyl-2,4,7-trioxo-1,2,3,4,7,8-hexahydropyrido[2,3-d]pyrimidin-5-yl)amino)phenyl)acetamide
品牌:毕得
BD450051871700-25-395%
登录 100mg
871700-18-4
1-Cyclopropyl-3-(2-fluoro-4-iodophenyl)urea
1-Cyclopropyl-3-(2-fluoro-4-iodophenyl)urea
品牌:毕得
BD244321871700-18-495%
登录 100mg
871700-26-4
2-Cyano-N-cyclopropyl-N-((2-fluoro-4-iodophenyl)carbamoyl)acetamide
2-Cyano-N-cyclopropyl-N-((2-fluoro-4-iodophenyl)carbamoyl)acetamide
品牌:毕得
BD244322871700-26-495%
登录 1g
871700-30-0
N'-(1-Cyclopropyl-3-(2-fluoro-4-iodophenyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)-N,N-dimethylformimidamide
N'-(1-Cyclopropyl-3-(2-fluoro-4-iodophenyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)-N,N-dimethylformimidamide
品牌:毕得
BD01661488871700-30-095%
登录 100mg
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