达克利司是咪唑喹啉衍生物, 是一种双重的 pan-class I PI3K 和 mTOR 抑制剂,作用于 p110α/γ/δ/β 和 mTOR,IC50 分别为 4 nM/5 nM/7 nM/75 nM 和 20.7 nM,抑制 mTORC1 和 mTORC2。

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723281-72-9
6-Bromo-4-chloro-3-nitroquinoline
6-Bromo-4-chloro-3-nitroquinoline
品牌:毕得
BD159709723281-72-997%
登录 1g 常备现货
115279-57-7
2-(4-Aminophenyl)-2-methylpropanenitrile
2-(4-Aminophenyl)-2-methylpropanenitrile
品牌:毕得
BD162094115279-57-797%
登录 5g 常备现货
853908-50-6
6-Bromo-3-nitroquinolin-4-ol
6-Bromo-3-nitroquinolin-4-ol
品牌:毕得
BD108453853908-50-697%
登录 10g 常备现货
71825-51-9
2-Methyl-2-(4-nitrophenyl)propanenitrile
2-Methyl-2-(4-nitrophenyl)propanenitrile
品牌:毕得
BD23853671825-51-997%
登录 25g 常备现货
915019-50-0
2-(4-(8-Bromo-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinolin-1-yl)phenyl)-2-methylpropanenitrile
2-(4-(8-Bromo-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinolin-1-yl)phenyl)-2-methylpropanenitrile
品牌:毕得
BD249830915019-50-095+%
登录 50mg
915019-51-1
2-(4-((6-Bromo-3-nitroquinolin-4-yl)amino)phenyl)-2-methylpropanenitrile
2-(4-((6-Bromo-3-nitroquinolin-4-yl)amino)phenyl)-2-methylpropanenitrile
品牌:毕得
BD234390915019-51-195+%
登录 1g
915019-52-2
2-(4-((3-Amino-6-bromoquinolin-4-yl)amino)phenyl)-2-methylpropanenitrile
2-(4-((3-Amino-6-bromoquinolin-4-yl)amino)phenyl)-2-methylpropanenitrile
品牌:毕得
BD234391915019-52-295+%
登录 1g
915019-53-3
2-(4-(8-Bromo-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinolin-1-yl)phenyl)-2-methylpropanenitrile
2-(4-(8-Bromo-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinolin-1-yl)phenyl)-2-methylpropanenitrile
品牌:毕得
BD234392915019-53-395%
登录 100mg
1