达鲁舍替是一种极光激酶 (aurora kinase) 抑制剂，能够抑制 Aurora A，Aurora B 和 Aurora C 的活性，IC50 值分别为 13，79 和 61 nM。
4-(4-Methylpiperazin-1-yl)benzoic acid
tert-Butyl 3-amino-4,6-dihydropyrrolo[3,4-c]pyrazole-5(1H)-carboxylate
(R)-(-)-alpha-Methoxyphenylacetic Acid
5-tert-Butyl 1-ethyl 3-aminopyrrolo[3,4-c]pyrazole-1,5(4H,6H)-dicarboxylate
Ethyl 3-(4-(4-methylpiperazin-1-yl)benzamido)-5,6-dihydropyrrolo[3,4-c]pyrazole-1(4H)-carboxylate
5-tert-Butyl 1-ethyl 3-(4-(4-methylpiperazin-1-yl)benzamido)pyrrolo[3,4-c]pyrazole-1,5(4H,6H)-dicarboxylate
