替米沙坦是一种有效的血管紧张素II 1型受体 (angiotensin II type 1 receptor) 拮抗剂，能够抑制其活性，IC50 值为 9.2 nM，用于高血压的治疗。
N-Methyl-1,2-benzenediamine dihydrochloride
Methyl 4-(butyrylamino)-3-methyl-5-nitrobenzoate
1,7'-Dimethyl-2'-propyl-1H,1'H-2,5'-bibenzo[d]imidazole
Methyl 4-butyramido-3-methylbenzoate
4-Bromo-2-methyl-6-nitroaniline
Methyl 4-amino-3-methylbenzoate
4-Methyl-2-propyl-1H-benzo[d]imidazole-6-carboxylic acid
2-Boc-4'-(Bromomethyl)biphenyl
Methyl 2-[4-(Bromomethyl)phenyl]benzoate
Methyl 4'-((1,7'-dimethyl-2'-propyl-1H,3'H-[2,5'-bibenzo[d]imidazol]-3'-yl)methyl)-[1,1'-biphenyl]-2-carboxylate
Methyl 7-methyl-2-propyl-1H-benzo[d]imidazole-5-carboxylate
Methyl 3-amino-4-butyramido-5-methylbenzoate
